Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50129409((R)-1-(3-Aminomethyl-pyrrolidin-1-yl)-2-((R)-3,3-d...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50129409((R)-1-(3-Aminomethyl-pyrrolidin-1-yl)-2-((R)-3,3-d...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity against human muscarinic acetylcholine receptor M3 in transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50129409((R)-1-(3-Aminomethyl-pyrrolidin-1-yl)-2-((R)-3,3-d...)
Affinity DataKi:  130nMAssay Description:Binding affinity against human muscarinic acetylcholine receptor M2 in transfected CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed