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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Ligand
BDBM22864
(2-[2-(3,3-diphenylpropyl)-1H-imidazol-4-yl]ethan-1...)
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Affinity Data
Ki: >1.00E+4nM ΔG°: >-29.7kJ/mole
pH: 7.4 T: 2°C
Assay Description:
Ligand displacement assays were performed on The SK-N-MC/hH4R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
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In Depth
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Article
PubMed
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Target
Histamine H1 receptor
(Homo sapiens (Human))
Vrije Universiteit Amsterdam
Curated by
ChEMBL
Ligand
BDBM22864
(2-[2-(3,3-diphenylpropyl)-1H-imidazol-4-yl]ethan-1...)
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Affinity Data
IC50: 794nM
Assay Description:
Inhibitory activity against human Histamine H1 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI