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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin B(Capra hircus (Goat))
Kurukshetra University

Curated by ChEMBL
LigandPNGBDBM50320734(4-Hydroxy-benzoic acid hydrazide | 4-hydroxybenzoh...)
Affinity DataKi:  1.90E+3nMAssay Description:Competitive inhibition of cathepsin B in goat liver using alpha-N-benzoyl-D,L-arginine-2-naphthylamide as substrate by colorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
King Saud University

Curated by ChEMBL
LigandPNGBDBM50320734(4-Hydroxy-benzoic acid hydrazide | 4-hydroxybenzoh...)
Affinity DataKi:  1.77E+5nMAssay Description:Inhibition of mashroom tyrosinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloperoxidase(Homo sapiens (Human))
University Sarajevo School Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50320734(4-Hydroxy-benzoic acid hydrazide | 4-hydroxybenzoh...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of MPO in human neutrophils using H2O2 as substrate measured after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50320734(4-Hydroxy-benzoic acid hydrazide | 4-hydroxybenzoh...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate preincubated for 15 mins followed by addition of subs...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed