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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mitogen-activated protein kinase kinase kinase kinase 4
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50011560
(CHEMBL3262579 | US9592235, Example 187 | US9855269...)
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Affinity Data
IC50: 60nM
Assay Description:
Inhibition of human MAP4K4 using 5-FAM-LGRDKYKTLRQIRQ-COOH as substrate by Z'-LYTE assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase kinase 4
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50011560
(CHEMBL3262579 | US9592235, Example 187 | US9855269...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 84nM
Assay Description:
The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase kinase 4
(Homo sapiens (Human))
Genentech
Curated by
ChEMBL
Ligand
BDBM50011560
(CHEMBL3262579 | US9592235, Example 187 | US9855269...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 84nM
Assay Description:
The kinase activity of purified human MAP4K4 kinase domain was measured by monitoring the phosphorylation of a peptide substrate derived from moesin ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI