Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-lipoxygenase(Bos taurus)
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50052459(10-(4-Amino-phenylsulfanyl)-1,8-dihydroxy-10H-anth...)
Affinity DataIC50:  7.00E+3nMAssay Description:Tested for inhibition of 5-lipoxygenase as inhibition of 5-HETE and LTB4 biosynthesis in bovine PMNLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid lipoxygenase ALOX12(Mus musculus)
UniversitäT Regensburg

Curated by ChEMBL
LigandPNGBDBM50052459(10-(4-Amino-phenylsulfanyl)-1,8-dihydroxy-10H-anth...)
Affinity DataIC50: >3.00E+4nMAssay Description:Tested for inhibition of 12-LO (12-lipoxygenase) as an inhibitor of 12(S)-HETE biosynthesis in mouse epidermal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed