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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50207492
(1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-cyclopenty...)
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Affinity Data
IC50: 39nM
Assay Description:
Inhibition of FLT3 by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50207492
(1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-cyclopenty...)
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Copy InChI
Affinity Data
IC50: 153nM
Assay Description:
Inhibition of VEGF-induced human KDR phosphorylation in mouse 3T3 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Punjabi University
Curated by
ChEMBL
Ligand
BDBM50207492
(1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-cyclopenty...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 850nM
Assay Description:
Inhibition of c-Kit by HTRF method
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Punjabi University
Curated by
ChEMBL
Ligand
BDBM50207492
(1-(4-(3-amino-1H-indazol-4-yl)phenyl)-3-cyclopenty...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 850nM
Assay Description:
Inhibition of c-Kit by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI