Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAdenosine receptor A2a(Homo sapiens (Human))
Universita Di Trieste

Curated by ChEMBL
LigandPNGBDBM50360186(CHEMBL1927446)
Affinity DataKi:  90.1nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Trieste

Curated by ChEMBL
LigandPNGBDBM50360186(CHEMBL1927446)
Affinity DataKi:  2.95E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universita Di Trieste

Curated by ChEMBL
LigandPNGBDBM50360186(CHEMBL1927446)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human recombinant adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase act...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed