Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 16 hits in this display
Ki: 0.0490nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
BDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
Ki: 1.5nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation countingMore data for this Ligand-Target Pair
BDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
Ki: 29nMAssay Description:Displacement of [3H]Naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
BDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
Ki: 29nMAssay Description:Displacement of [3H]naltrindole from human delta-opioid receptor expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
EC50: 73nMAssay Description:Agonist activity at human mu opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation countingMore data for this Ligand-Target Pair
BDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
BDBM50143602(20-cyclopropylmethyl-(1R,12R)-7-thia-5,20-diazapen...)
EC50: 2.40nMAssay Description:Agonist activity at human kappa opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by scintillation countingMore data for this Ligand-Target Pair