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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
NEDD8-conjugating enzyme UBE2F
(Homo sapiens (Human))
Taiho Pharmaceutical
US Patent
Ligand
BDBM321040
(4-Amino-5-[2-[2,6-difluoro-4-[(3R)-3-hydroxypyrrol...)
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Affinity Data
IC50: 4.30nM
Assay Description:
A purified NAE (heterodimer of APPBP1 and UBA3) solution was prepared in the following manner. The human APPBP1 gene (NCBI Reference Sequence number:...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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Target
Carbonic anhydrase 2
(Homo sapiens (Human))
Taiho Pharmaceutical
US Patent
Ligand
BDBM321040
(4-Amino-5-[2-[2,6-difluoro-4-[(3R)-3-hydroxypyrrol...)
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Copy InChI
Affinity Data
IC50: >1.00E+3nM
Assay Description:
The carbonic anhydrase II enzyme activity inhibition was measured by measuring the esterase activity in which carbonic anhydrase II degrades 4-nitrop...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Carbonic anhydrase 2
(Homo sapiens (Human))
Taiho Pharmaceutical
US Patent
Ligand
BDBM321040
(4-Amino-5-[2-[2,6-difluoro-4-[(3R)-3-hydroxypyrrol...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+3nM
Assay Description:
The carbonic anhydrase II enzyme activity inhibition was measured by measuring the esterase activity in which carbonic anhydrase II degrades 4-nitrop...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI