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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNEDD8-conjugating enzyme UBE2F(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM320987(4-Amino-5-[2-(2-cyanophenyl)ethynyl]-7-[(2R,3R,4S,...)
Affinity DataIC50:  18nMAssay Description:A purified NAE (heterodimer of APPBP1 and UBA3) solution was prepared in the following manner. The human APPBP1 gene (NCBI Reference Sequence number:...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM320987(4-Amino-5-[2-(2-cyanophenyl)ethynyl]-7-[(2R,3R,4S,...)
Affinity DataIC50: >1.00E+3nMAssay Description:The carbonic anhydrase II enzyme activity inhibition was measured by measuring the esterase activity in which carbonic anhydrase II degrades 4-nitrop...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM320987(4-Amino-5-[2-(2-cyanophenyl)ethynyl]-7-[(2R,3R,4S,...)
Affinity DataIC50: >1.00E+3nMAssay Description:The carbonic anhydrase II enzyme activity inhibition was measured by measuring the esterase activity in which carbonic anhydrase II degrades 4-nitrop...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent