Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 22 hits in this display
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
Ki: 9.30nMAssay Description:Inhibition of Sprague-Dawley rat brain cytosolic Adk using [2-3H]adenosine incubated for 15 mins by scintillation spectrometryMore data for this Ligand-Target Pair
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
IC50: 7.00E+3nMAssay Description:Inhibition of DOT1L (unknown origin) using chicken nucleosome as substrate in presence of [3H]SAM incubated for 1 hr by TopCount methodMore data for this Ligand-Target Pair
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)
BDBM50375654(CHEMBL99203 | US11633415, Compound 5-iodotubercidi...)