Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095366(5-(2-Bromo-benzyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  0.170nMAssay Description:Inhibitory activity against cytosolic adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50095366(5-(2-Bromo-benzyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataIC50:  33nMAssay Description:Inhibitory activity against intact cell adenosine kinase by ADO phosphorylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed