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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

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TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50310345(6-(3-amino-1-(3-(2-oxoindolin-6-yl)phenyl)-1H-pyra...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human MK2 by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed