Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50298552(5-[(4-Biphenylmethyl)carbonyl]amino-8-(2-phenyleth...)
Affinity DataKi:  46.9nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50298552(5-[(4-Biphenylmethyl)carbonyl]amino-8-(2-phenyleth...)
Affinity DataKi:  84.3nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50298552(5-[(4-Biphenylmethyl)carbonyl]amino-8-(2-phenyleth...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50298552(5-[(4-Biphenylmethyl)carbonyl]amino-8-(2-phenyleth...)
Affinity DataIC50:  1.11E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced adenylyl cyclase activityChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed