Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 1 hits in this display
BDBM50305027((6-(cyclohexylamino)pyridin-3-yl)(piperidin-1-yl)m...)
IC50: >1.00E+4nMAssay Description:Antagonist activity at human mGluR5 assessed as inhibition of glutamate-induced elevation of intracellular calcium concentrationMore data for this Ligand-Target Pair