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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Monoglyceride lipase
(Homo sapiens (Human))
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50394369
(CHEMBL2159781)
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Affinity Data
Ki: 75.7nM
Assay Description:
Irreversible inhibition of human MAGL using p-nitrophenylpropionate as substrate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Monoglyceride lipase
(Homo sapiens (Human))
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50394369
(CHEMBL2159781)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.540nM
Assay Description:
Inhibition of human MAGL assessed as [3H]-2-OG hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liquid scintil...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Fatty-acid amide hydrolase 1
(Homo sapiens (Human))
Sapienza University Of Rome
Curated by
ChEMBL
Ligand
BDBM50394369
(CHEMBL2159781)
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Copy InChI
Affinity Data
IC50: 562nM
Assay Description:
Inhibition of human recombinant FAAH assessed as [3H]-AEA hydrolysis preincubated for 30 mins before [3H]-2-OG addition measured after 10 mins by liq...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI