Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi:  2.30nM ΔG°:  -48.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi:  130nM ΔG°:  -38.9kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi: >2.00E+3nM ΔG°: >-32.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi:  6.90E+3nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Wyeth Research

LigandPNGBDBM28579(1-sulfonylindazole, 7a | N-[1-(naphthalene-1-sulfo...)
Affinity DataKi:  8.50E+3nM ΔG°:  -28.7kJ/molepH: 7.4 T: 2°CAssay Description:Competition experiments were performed in the presence radioligand with membrane protein (obtained from cells expressing the receptor) and test compo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed