Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Adenosine receptor A3
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50254611
(CHEMBL519614 | N-(2-phenyl-2H-pyrazolo[3,4-c]quino...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 10.5nM
Assay Description:
Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cells by scintillation counting
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A3
(Homo sapiens (Human))
Università
Curated by
ChEMBL
Ligand
BDBM50254611
(CHEMBL519614 | N-(2-phenyl-2H-pyrazolo[3,4-c]quino...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 76nM
Assay Description:
Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP accumulati...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI