Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50254611(CHEMBL519614 | N-(2-phenyl-2H-pyrazolo[3,4-c]quino...)
Affinity DataKi:  10.5nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50254611(CHEMBL519614 | N-(2-phenyl-2H-pyrazolo[3,4-c]quino...)
Affinity DataIC50:  76nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed