Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 33 hits in this display
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50175570((S)-1-Phenyl-3,4-dihydro-1H-isoquinoline-2-carboxy...)
BDBM50344284(CHEMBL1200803 | Solifenacin | Solifenacin succinat...)
IC50: 63.5nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
BDBM50344284(CHEMBL1200803 | Solifenacin | Solifenacin succinat...)
IC50: 131nMAssay Description:Displacement of [3H]NMS from human muscarinic M3 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
BDBM50344284(CHEMBL1200803 | Solifenacin | Solifenacin succinat...)
IC50: 574nMAssay Description:Displacement of [3H]NMS from human muscarinic M2 receptor expressed in CHO-K1 cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
IC50: 4.30E+3nMAssay Description:Inhibition of Cav1.2 current measured using QPatch automatic path clamp system in CHO cells expressing Cav1.2, beta-2 and alpha-2/delta-1 subunitsMore data for this Ligand-Target Pair