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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Muscarinic acetylcholine receptor M1
(RAT)
Astellas Pharma
Curated by
ChEMBL
Ligand
BDBM50175574
((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
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Affinity Data
Ki: 0.950nM
Assay Description:
Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M3
(RAT)
Astellas Pharma
Curated by
ChEMBL
Ligand
BDBM50175574
((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.5nM
Assay Description:
Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M1
(RAT)
Astellas Pharma
Curated by
ChEMBL
Ligand
BDBM50175574
((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 8.30nM
Assay Description:
Binding affinity for rat cortex muscarinic acetylcholine receptor M1 using [3H]pirenzepine
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(RAT)
Astellas Pharma
Curated by
ChEMBL
Ligand
BDBM50175574
((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 15nM
Assay Description:
Binding affinity for rat heart muscarinic acetylcholine receptor M2 using [3H]quinuclidinyl benzilate
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M3
(RAT)
Astellas Pharma
Curated by
ChEMBL
Ligand
BDBM50175574
((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 21nM
Assay Description:
Binding affinity for rat salivary gland muscarinic acetylcholine receptor M3 using [3H]N-methylscopolamine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(RAT)
Astellas Pharma
Curated by
ChEMBL
Ligand
BDBM50175574
((S)-1-Thiophen-3-yl-3,4-dihydro-1H-isoquinoline-2-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 110nM
Assay Description:
Binding affinity for rat heart muscarinic acetylcholine receptor M2 using [3H]quinuclidinyl benzilate
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI