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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Sigma non-opioid intracellular receptor 1
(Homo sapiens (Human))
Albany Molecular Research
Curated by
ChEMBL
Ligand
BDBM50038705
(1-Phenyl-cyclopentanecarboxylic acid 2-(4-phenyl-p...)
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Affinity Data
Ki: 4nM
Assay Description:
Affinity at sigma-1 site by inhibition of [3H](+)-pentazocine (PENT) binding in guinea pig brain
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Muscarinic acetylcholine receptor M1
(RAT)
Albany Molecular Research
Curated by
ChEMBL
Ligand
BDBM50038705
(1-Phenyl-cyclopentanecarboxylic acid 2-(4-phenyl-p...)
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Copy InChI
Affinity Data
Ki: 170nM
Assay Description:
Binding affinity was measured as selectivity for sigma-1 site over muscarinic (M1) receptor in rat using [3H]pirenzepine as radioligand
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI