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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50143655(8-[2-(4-Phenyl-piperidin-1-yl)-ethyl]-8-aza-spiro[...)
Affinity DataKi:  3.66nMAssay Description:Binding affinity to the adrenergic receptor alpha-1D of rat aortaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50143655(8-[2-(4-Phenyl-piperidin-1-yl)-ethyl]-8-aza-spiro[...)
Affinity DataKi:  25.9nMAssay Description:Binding affinity to human 5-hydroxytryptamine 1A receptor was measured using [3H]-8-hydroxy-2-(di-n-propylamine) tetraline [3H]-8-OH-DPAT) as radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Recordati

Curated by ChEMBL
LigandPNGBDBM50143655(8-[2-(4-Phenyl-piperidin-1-yl)-ethyl]-8-aza-spiro[...)
Affinity DataKi:  274nMAssay Description:Binding affinity constant against alpha-1B adrenergic receptor of guinea pig spleenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Recordati

Curated by ChEMBL
LigandPNGBDBM50143655(8-[2-(4-Phenyl-piperidin-1-yl)-ethyl]-8-aza-spiro[...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor through displacement of [3H]-prazosin in epididymal rat vas deferens.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed