Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50074004(1'-[2-(2-pyridyl)ethyl]spiro[3,4-dihydro-2H-chrome...)
Affinity DataKi:  793nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1C adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50074004(1'-[2-(2-pyridyl)ethyl]spiro[3,4-dihydro-2H-chrome...)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1B adrenergic receptor expressed in LM cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50074004(1'-[2-(2-pyridyl)ethyl]spiro[3,4-dihydro-2H-chrome...)
Affinity DataKi:  1.52E+3nMAssay Description:Displacement of [125I]-HEAT from human Alpha-1D adrenergic receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed