Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(RAT)
University Of Uppsala

Curated by ChEMBL

LigandBDBM50230003(CHEMBL97890)Copy SMILESCopy InChI

Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
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TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
University Of Uppsala

Curated by ChEMBL

LigandBDBM50230003(CHEMBL97890)Copy SMILESCopy InChI

Affinity DataKd:  8.10E+3nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaantibodypediaantibodypediaantibodypediaantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidPatents

In DepthDetails ArticlePubMed
Copy BDB DOI