Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 1(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50204432(6-benzyloxy-2,3,4,4a,9,9a-hexahydro-beta-carbolin-...)
Affinity DataIC50:  1.67E+3nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of intracellular calcium ion mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed