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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Nociceptin receptor
(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by
ChEMBL
Ligand
BDBM50204780
(8-cyclohexylmethyl-1-phenyl-1,3,8-triaza-spiro[4.5...)
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Affinity Data
Ki: 61nM
Assay Description:
Displacement of [125I]nociceptin from human nociceptin receptor expressed in CHO cell membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kappa-type opioid receptor
(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by
ChEMBL
Ligand
BDBM50204780
(8-cyclohexylmethyl-1-phenyl-1,3,8-triaza-spiro[4.5...)
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Affinity Data
Ki: 517nM
Assay Description:
Displacement of [3H]diprenorphine from human kappa opioid receptor expressed in CHO cell membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by
ChEMBL
Ligand
BDBM50204780
(8-cyclohexylmethyl-1-phenyl-1,3,8-triaza-spiro[4.5...)
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Affinity Data
Ki: 887nM
Assay Description:
Displacement of [3H]diprenorphine from human mu opioid receptor expressed in CHO cell membrane
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by
ChEMBL
Ligand
BDBM50204780
(8-cyclohexylmethyl-1-phenyl-1,3,8-triaza-spiro[4.5...)
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Copy InChI
Affinity Data
Ki: 7.37E+4nM
Assay Description:
Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cell membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI