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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Leukotriene A-4 hydrolase
(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical
Ligand
BDBM24235
(3-(1-{[4-(1,3-benzothiazol-2-yloxy)phenyl]methyl}p...)
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Affinity Data
IC50: 10nM
T: 2°C
Assay Description:
Recombinant human LTA4H was incubated with various concentrations of test compound for 10 min at room temperature in assay buffer, and the substrate,...
More data for this Ligand-Target Pair
Target Info
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KEGG
UniProtKB/SwissProt
B.MOAD
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antibodypedia
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Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical
Ligand
BDBM24235
(3-(1-{[4-(1,3-benzothiazol-2-yloxy)phenyl]methyl}p...)
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Affinity Data
IC50: 2.40E+4nM
Assay Description:
Compounds were assessed for their ability to displace [3H]astemizole using membranes from HEK-293 cells expressing the hERG K+ channel.
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
UniProtKB/TrEMBL
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI