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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetLeukotriene A-4 hydrolase(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical

LigandPNGBDBM24235(3-(1-{[4-(1,3-benzothiazol-2-yloxy)phenyl]methyl}p...)
Affinity DataIC50:  10nMT: 2°CAssay Description:Recombinant human LTA4H was incubated with various concentrations of test compound for 10 min at room temperature in assay buffer, and the substrate,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical

LigandPNGBDBM24235(3-(1-{[4-(1,3-benzothiazol-2-yloxy)phenyl]methyl}p...)
Affinity DataIC50:  2.40E+4nMAssay Description:Compounds were assessed for their ability to displace [3H]astemizole using membranes from HEK-293 cells expressing the hERG K+ channel.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed