Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50425110(CHEMBL2312927)
Affinity DataIC50:  140nMAssay Description:Inhibition of human Kv1.5 channel expressed in CHO cells by high throughput planar patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50425110(CHEMBL2312927)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of IK channel (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed