Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50277017(4-(naphthalen-1-ylsulfonyl)-2-(piperazin-1-yl)benz...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptor expressed in human HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50277017(4-(naphthalen-1-ylsulfonyl)-2-(piperazin-1-yl)benz...)
Affinity DataIC50:  96nMAssay Description:Antagonist activity at human cloned 5HT6 receptor expressed in human HeLa cells assessed as blockage of 5HT-stimulated cAMP formation after 10 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed