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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandPNGBDBM50208259(CHEMBL3884704)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-LSD from human recombinant 5-HT6 receptor expressed in CHOK1 cell membranes measured after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandPNGBDBM50208259(CHEMBL3884704)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of equine serum BuChE preincubated for 5 mins followed by butyrylthiocholine iodide substrate addition measured after 5 mins by Ellman's m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Jagiellonian University Collegium Medicum

Curated by ChEMBL
LigandPNGBDBM50208259(CHEMBL3884704)
Affinity DataIC50:  4.41E+3nMAssay Description:Inhibition of electric eel AChE preincubated for 5 mins followed by acetylthiocholine iodide substrate addition measured after 5 mins by Ellman's met...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed