Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50218176((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-4-yl)thia...)Copy SMILESCopy InChI

Affinity DataKi:  97nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50218176((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-4-yl)thia...)Copy SMILESCopy InChI

Affinity DataEC50:  65nMAssay Description:Agonist activity at human adrenergic beta-3 receptor expressed in CHO cells assessed as cAMP productionMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI