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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50089458(4-[5-(3-Cyclopentyl-propyl)-[1,2,4]oxadiazol-3-yl]...)
Affinity DataIC50:  962nMAssay Description:Binding affinity towards Beta-2 adrenergic receptor prepared from CHO cells expressing the cloned human receptor in the presence of [125I]-iodocyanop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50089458(4-[5-(3-Cyclopentyl-propyl)-[1,2,4]oxadiazol-3-yl]...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity towards cloned human Beta-1 adrenergic receptor prepared from CHO cells in the presence of [125I]-iodocyanopindololMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50089458(4-[5-(3-Cyclopentyl-propyl)-[1,2,4]oxadiazol-3-yl]...)
Affinity DataEC50:  15nMAssay Description:Agonist activity as increasedn cAMP production in Chinese hamster ovary (CHO)cells expressing human beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed