Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetProtein kinase C alpha type(Homo sapiens (Human))
Virginia Polytechnic Institute And State University

Curated by ChEMBL
LigandPNGBDBM50269516(CHEMBL518414 | Calceolarioside B)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan Normal University

Curated by ChEMBL
LigandPNGBDBM50269516(CHEMBL518414 | Calceolarioside B)
Affinity DataIC50:  3.53E+4nMAssay Description:Inhibition of aromatase preincubated with 2.6 mM NADP+ for 10 mins before substrate addition measured after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed