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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAldo-keto reductase family 1 member B1(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50362657(CHEMBL1939430)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of rat lens aldose reductase using DL-glyceraldehyde as substrate after 30 mins by fluorescence microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50362657(CHEMBL1939430)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of alpha-glucosidase activity of maltase in rat small intestinal brush border membrane fraction using maltose as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50362657(CHEMBL1939430)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibition of alpha-glucosidase activity of sucrase in rat small intestinal brush border membrane fraction using maltose as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed