Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Evotec Internatonal

US Patent
LigandPNGBDBM289126(US10093660, Example 1.7)
Affinity DataIC50:  2nMT: 2°CAssay Description:ASSAY SETUP: The inhibition of kinase activity of MNK2a was assessed using pre-activated GST-MNK2a. The white, 384-well OptiPlate F plates were purch...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec Internatonal

US Patent
LigandPNGBDBM289126(US10093660, Example 1.7)
Affinity DataIC50:  18nMAssay Description:MNK1 Data can be obtained from the MNK1 Z′-LYTEŽ assay. The MNK1 Z′-LYTEŽ screening protocol and assay conditions are also described on w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Evotec Internatonal

US Patent
LigandPNGBDBM289126(US10093660, Example 1.7)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Mnk2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Evotec Internatonal

US Patent
LigandPNGBDBM289126(US10093660, Example 1.7)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Mnk1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed