Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMuscarinic acetylcholine receptor M1(RAT)
Hoffmann-La Roche

US Patent

LigandBDBM261726(4-(4-chlorobenzyl)- 1-fluoro-N- ((3RS,4SR)-3- hydr...)Copy SMILESCopy InChI

Affinity DataEC50:  273nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair

Target InfoReactome pathwayKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent

LigandBDBM261726(4-(4-chlorobenzyl)- 1-fluoro-N- ((3RS,4SR)-3- hydr...)Copy SMILESCopy InChI

Affinity DataEC50:  152nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI