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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetBeta-lactamase(Escherichia coli)
Northwestern University Medical School

Curated by ChEMBL
LigandPNGBDBM50067891(5-chlorothiophen-2-ylboronic acid | 5-chlorothiphe...)
Affinity DataKi:  410nMAssay Description:Inhibitory activity against E. coli AmpC beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Escherichia coli)
Northwestern University Medical School

Curated by ChEMBL
LigandPNGBDBM50067891(5-chlorothiophen-2-ylboronic acid | 5-chlorothiphe...)
Affinity DataIC50:  2.00E+3nMAssay Description:Compound was tested for its specificity against AmpC beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Tokushima University

Curated by ChEMBL
LigandPNGBDBM50067891(5-chlorothiophen-2-ylboronic acid | 5-chlorothiphe...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human DAO using D-serine as substrate after 20 mins in presence of FADMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Northwestern University Medical School

Curated by ChEMBL
LigandPNGBDBM50067891(5-chlorothiophen-2-ylboronic acid | 5-chlorothiphe...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was tested for its specificity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin-2(Homo sapiens (Human))
Northwestern University Medical School

Curated by ChEMBL
LigandPNGBDBM50067891(5-chlorothiophen-2-ylboronic acid | 5-chlorothiphe...)
Affinity DataIC50: >2.00E+5nMAssay Description:Compound was tested for its specificity against beta-trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed