Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271701(2,6-bis(3-carboxyacrylamido)benzoic acid | 4,4'-(2...)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at LPA3 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271701(2,6-bis(3-carboxyacrylamido)benzoic acid | 4,4'-(2...)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271701(2,6-bis(3-carboxyacrylamido)benzoic acid | 4,4'-(2...)
Affinity DataIC50:  355nMAssay Description:Antagonist activity at LPA2 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophosphatidic acid receptor 2(Homo sapiens (Human))
The University Of Memphis

Curated by ChEMBL
LigandPNGBDBM50271701(2,6-bis(3-carboxyacrylamido)benzoic acid | 4,4'-(2...)
Affinity DataIC50:  355nMAssay Description:Antagonist activity at LPA2 receptor (unknown origin) expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium conce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed