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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNeprilysin(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50006115((R)-RETRO-THIORPHAN | (RETRO)N-(1-Mercaptomethyl-2...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of NEP 24.11 (unknown origin) by fluorometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50006115((R)-RETRO-THIORPHAN | (RETRO)N-(1-Mercaptomethyl-2...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibitory constant against thermolysin.More data for this Ligand-Target Pair
TargetNeprilysin(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006115((R)-RETRO-THIORPHAN | (RETRO)N-(1-Mercaptomethyl-2...)
Affinity DataIC50:  210nMAssay Description:Concentration for 50% inhibition of activity of rat kidney enkephalinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50006115((R)-RETRO-THIORPHAN | (RETRO)N-(1-Mercaptomethyl-2...)
Affinity DataIC50:  1.00E+9nMAssay Description:Inhibition of angiotensin I converting enzyme in silicoMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed