Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetSolute carrier family 22 member 2(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataIC50:  7.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 1(RAT)
Institute Of Anatomy Of The Bayerische Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataIC50:  7.40E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 10 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Zhengzhou University

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataIC50:  8.00E+5nMAssay Description:Inhibition of KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to human PHD2-Mn(II) using 12.5% H2O/87.5% D2O MQC spectrometer operated at 500 MHz at 298K temperature in presence of HIF1alpha (55...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataKd:  900nMAssay Description:Binding affinity to human PHD2 catalytic domain (181 to 426) Mn2 expressed in Escherichia coli by 1H-15N HSQC titration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataKd:  900nMAssay Description:Binding affinity to human PHD2-Mn(II) using 12.5% H2O/87.5% D2O MQC spectrometer operated at 500 MHz at 298K temperatureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to human PHD2-Mn(II) using 12.5% H2O/87.5% D2O MQC spectrometer operated at 500 MHz at 313K temperatureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human PHD2-Mn(II) using 100% H2O MQC spectrometer operated at 23 MHz at 313K temperatureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEgl nine homolog 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50303766(2-oxoglutaric acid | 2-oxopentanedioic acid | CHEM...)
Affinity DataKd:  900nMAssay Description:Binding affinity to human PHD2 by nondenaturing ESI-MSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed