Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM50065771(4-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]qui...)
BDBM50065771(4-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]qui...)
BDBM50065771(4-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]qui...)
Ki: 81.3nMAssay Description:Binding affinity at cloned human adenosine A3 receptor expressed in HEK-293 cells was determined using [125I]-AB-MECA as radioligandMore data for this Ligand-Target Pair
BDBM50065771(4-(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]qui...)
IC50: 1.90E+3nMAssay Description:Inhibition of 50 uM 5`-(N-ethylcarboxamido)adenosine induced cAMP production in CHO cell line expressing human Adenosine A2B receptor at 50 uMMore data for this Ligand-Target Pair