Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetHistamine H1 receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416669(CHEMBL1222553)
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at human recombinant histamine H1 receptor expressed in CHO cells by FLPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416669(CHEMBL1222553)
Affinity DataKi:  316nMAssay Description:Antagonist activity at human 5HT2A receptor expressed in HEK cells assessed as intracellular calcium luminescence by aequorin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416669(CHEMBL1222553)
Affinity DataKi: >794nMAssay Description:Antagonist activity at human 5HT2C receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50416669(CHEMBL1222553)
Affinity DataKi: >794nMAssay Description:Antagonist activity at human 5HT2B receptor expressed in human SHSY5Y cells by FLPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed