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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMonocarboxylate transporter 4(Homo sapiens (Human))
Institut De Recherche Exp£Rimentale Et Clinique (Irec)

Curated by ChEMBL
LigandPNGBDBM50442717(CHEMBL2442515)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of MCT4-mediated [14C]-lactate uptake in human SiHa cells in lactate-containing medium assessed as remaining lactate concentration in cult...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed