Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories

Curated by ChEMBL

LigandBDBM50095672(CHEMBL148129 | N-(1-Cycloheptylmethyl-piperidin-4-...)Copy SMILESCopy InChI

Affinity DataKi:  12nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M3 expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories

Curated by ChEMBL

LigandBDBM50095672(CHEMBL148129 | N-(1-Cycloheptylmethyl-piperidin-4-...)Copy SMILESCopy InChI

Affinity DataKi:  200nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M1 expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories

Curated by ChEMBL

LigandBDBM50095672(CHEMBL148129 | N-(1-Cycloheptylmethyl-piperidin-4-...)Copy SMILESCopy InChI

Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M2 expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI