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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Nanjing University
Ligand
BDBM167947
(1-(4-(3-Chlorophenyl)piperazin-1-yl)-3-(quinazolin...)
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Affinity Data
IC50: 47.4nM
pH: 7.2 T: 2°C
Assay Description:
VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Platelet-derived growth factor receptor beta
(Homo sapiens (Human))
Nanjing University
Ligand
BDBM167947
(1-(4-(3-Chlorophenyl)piperazin-1-yl)-3-(quinazolin...)
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Copy InChI
Affinity Data
IC50: 209nM
pH: 7.2 T: 2°C
Assay Description:
VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Fibroblast growth factor 2
(Homo sapiens (Human))
Nanjing University
Ligand
BDBM167947
(1-(4-(3-Chlorophenyl)piperazin-1-yl)-3-(quinazolin...)
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Copy InChI
Affinity Data
IC50: 402nM
pH: 7.2 T: 2°C
Assay Description:
VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Nanjing University
Ligand
BDBM167947
(1-(4-(3-Chlorophenyl)piperazin-1-yl)-3-(quinazolin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 413nM
pH: 7.2 T: 2°C
Assay Description:
VEGFR kinase assays were set up to assess the level of autophosphorylation based on DELFIA/Time-Resolved Fluorometry. 96-well plates were coated at r...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI