Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSucrase-isomaltase, intestinal(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024126(1-Hydroxymethyl-5-[(pyridin-3-ylmethyl)-amino]-cyc...)
Affinity DataIC50:  15nMAssay Description:Alpha-D-glucosidase inhibitory activity and enzyme inhibition in vitro against porcine sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50024126(1-Hydroxymethyl-5-[(pyridin-3-ylmethyl)-amino]-cyc...)
Affinity DataIC50:  330nMAssay Description:Inhibitory activity against porcine maltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed