Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat intestinal isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  640nMAssay Description:Inhibition of rat isomaltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of rat intestinal sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of rat sucraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 mins by glucose-oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysosomal alpha-glucosidase(Rattus norvegicus)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of rat intestinal maltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMaltase-glucoamylase(Homo sapiens (Human))
Kindai University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human intestinal maltase using maltose as substrate incubated for 30 mins and immediately heated for 2 mins by glucose oxidase methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSucrase-isomaltase, intestinal(Rattus norvegicus (Rat))
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat intestinal maltaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen debranching enzyme(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50338669(CHEMBL1684162 | Neosalacinol)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of amylo-1,6-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed