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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetAurora kinase B(Homo sapiens (Human))
Konkuk University

LigandPNGBDBM153265(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-3-[(2S,3R,4S...)
Affinity DataIC50:  1.07E+4nMAssay Description:The kinase assay was performed using the EMD Millipore KinaseProfiler service assay protocol. Aurora B kinase was supplied by EMD Millipore Corp. The...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Homo sapiens (Human))
Catholic University Of Daegu

LigandPNGBDBM153265(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-3-[(2S,3R,4S...)
Affinity DataIC50:  8.48E+4nMpH: 8.0 T: 2°CAssay Description:Briefly, 140 μL of sodium phosphate buffer (pH 8.0), 20 μL of each tested compound with different concentrations (4, 20, and 100 μM) a...More data for this Ligand-Target Pair
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TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Catholic University Of Daegu

LigandPNGBDBM153265(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-3-[(2S,3R,4S...)
Affinity DataIC50:  1.00E+5nMpH: 6.0Assay Description:PTP1B activity was measured by adding 2mM p-NPP and PTP1B in a 50 mM citrate buffer (pH 6.0, 0.1 M NaCl, 1 mMEDTA, and 1 mM dithiothreitol), with or ...More data for this Ligand-Target Pair
In DepthDetails