Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetType 1 fimbrin D-mannose specific adhesin(Escherichia coli (strain K12))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347465(CHEMBL1802185)
Affinity DataIC50:  6.70nMAssay Description:Competitive inhibition of His-tagged FimH carbohydrate recognizing domain expressed in Escherichia coli HM125 using ABTS-substrate after 3 hrs by cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType 1 fimbiral adhesin FimH(Escherichia coli (strain UTI89 / UPEC))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50347465(CHEMBL1802185)
Affinity DataIC50:  1.00E+4nMAssay Description:Antagonist activity at Escherichia coli UT189 FimH in guinea pig red blood cells assessed as disaggregation of bacteria after 600 secs by aggregometr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage mannose receptor 1(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50399360(CHEMBL1852052)
Affinity DataIC50:  1.00E+6nMAssay Description:Displacement of biotinylated-TM PAA from human MMR after 3 hrs by colorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-type lectin domain family 4 member K(Homo sapiens (Human))
University Of Basel

Curated by ChEMBL
LigandPNGBDBM50399360(CHEMBL1852052)
Affinity DataIC50:  1.00E+6nMAssay Description:Displacement of biotinylated-TM PAA from human langerin after 3 hrs by colorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed