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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Array Biopharma
Curated by
ChEMBL
Ligand
BDBM120092
(US8697715, 14 | US9259470, 14)
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Affinity Data
Ki: 1.70nM
Assay Description:
Inhibition of 6-His tagged human ERK2 expressed in Escherichia coli measured over 30 mins by competition assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Array Biopharma
Curated by
ChEMBL
Ligand
BDBM120092
(US8697715, 14 | US9259470, 14)
Copy SMILES
Copy InChI
Affinity Data
IC50: 15.6nM
pH: 7.3
Assay Description:
Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Array Biopharma
Curated by
ChEMBL
Ligand
BDBM120092
(US8697715, 14 | US9259470, 14)
Copy SMILES
Copy InChI
Affinity Data
IC50: 15.6nM
pH: 7.3
Assay Description:
Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI